As modulator compoun... 申请号:JP2018009384 专利类型:发明授权 公开(公告)日:2018-01-24
状态:寻求转化 转让价格:面议
The present invention encompasses compounds of the formula (I) wherein the variables are defined herein which are suitable for the modulation of RORy and the treatment of diseases related to the mo...
As inhibitor of spir... 申请号:JP2017502166 专利类型:发明授权 公开(公告)日:
状态:寻求转化 转让价格:面议
The present invention provides compounds of Formula (I) : or stereoisomers, tautomers, or pharmaceutically-acceptable salts thereof, wherein all the variables are as defined herein. These compound...
As inhibitor of TAFI... 申请号:JP2016517597 专利类型:发明授权 公开(公告)日:2014-06-05
状态:寻求转化 转让价格:面议
The present invention relates to macrocydic urea derivatives of the formula I (I) in which R1, R2, R3, V and Y are as defined below. The compounds of the formula I are inhibitors of the enzyme TAFI...
As inhibitor compoun... 申请号:JP2018550711 专利类型:发明申请 公开(公告)日:
状态:寻求转化 转让价格:面议
or pharmaceutically acceptable salts thereof, which are inhibitors of TAM kinases which are useful for the treatment of disorders such as cancer.
As inhibitor antidep... 申请号:JP2018562088 专利类型:发明申请 公开(公告)日:
状态:寻求转化 转让价格:面议
The present invention provides compounds of Formula (I) : or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compound...
As inhibitor ROCK [.... 申请号:JP2018536481 专利类型:发明申请 公开(公告)日:
状态:寻求转化 转让价格:面议
The present invention provides compounds of Formula (I) : or stereoisomers, tautomers, or pharmaceutically-acceptable salts thereof, wherein all the variables are as defined herein. These compound...
As inhibitor LRRK2 [... 申请号:JP2016508109 专利类型:发明授权 公开(公告)日:2014-04-14
状态:寻求转化 转让价格:面议
The present invention is directed to arylpyrrolopyridine derivatives of formula (A) The compounds are considered useful for the treatment of diseases associated with LRRK2 such as Lewy body dementia, ...
As heterocyclic sulf... 申请号:JP2016562466 专利类型:发明授权 公开(公告)日:2015-01-05
状态:寻求转化 转让价格:面议
Described are RORγ modulators of the formula (I), [INSERT CHEMICAL STRUCTURE HERE] or stereoisomers, tautomers, pharmaceutically acceptable salts, solvates, or prodrugs thereof, wherein all subs...
As hairpin peptide m... 申请号:JP2016543043 专利类型:发明授权 公开(公告)日:
状态:寻求转化 转让价格:面议
β-Hairpin peptidomimetics of the general formula cyclo(-Xaa1-Xaa2-Thr3-Xaa4-Ser5-Xaa6-Xaa7-Xaa8-Xaa9-Xaa10-Xaa11-Xaa12-Xaa13-) and pharmaceutically acceptable salts thereof, with Xaa1, Xaa2, Xaa4, ...
As gamma modulator c... 申请号:JP2018537810 专利类型:发明申请 公开(公告)日:2017-01-18
状态:寻求转化 转让价格:面议
The present invention encompasses compounds of the formula (I), wherein the variables are defined herein which are suitable for the modulation of RORγ and the treatment of diseases related to the mod...