专利名称 | MMP ACTIVATED VASCULAR DISRUPTING AGENTS | ||
申请号 | EP18194638 | 申请日 | |
公开(公告)号 | EP3446715A1 | 公开(公告)日 | 2009-10-20 |
申请(专利权)人 | 发明人 | FALCONER Robert Andrew; GILL Jason; ATKINSON Jennifer; LOADMAN Paul; BIBBY Michael; PATTERSON Laurence | |
专利来源 | 国家知识产权局 | 转化方式 | |
摘要 |
The present invention relates to prodrugs of vascular disrupting agents comprising a vascular disrupting agent (VDA) associated with a MMP proteolytic cleavage site and to the use of such prodrugs in the targeted treatment of cancer. |
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