专利名称 | SELECTIVE MAO-B INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF | ||
申请号 | JP2018166454 | 申请日 | |
公开(公告)号 | JP2019031495A | 公开(公告)日 | 2018-09-05 |
申请(专利权)人 | 发明人 | EDWARD EWALD PUTNINS; DAVID SCOTT GRIERSON; RONAN F B GEALAGEAS; ALICE ANDREE VALENTINE DEVINEAU; EDITH MARY DULLAGHAN | |
专利来源 | 国家知识产权局 | 转化方式 | |
摘要 |
PROBLEM TO BE SOLVED : To provide a series of compounds used in MAO inhibition. SOLUTION : There is provided a compound having the following formula. A1 and A2 are F, Cl, Br, CN, OMe, NO2, CO2H; E1 is ; E2 is H; D is H, Me, CH2Cl, CH2F, CH2Br, CH2I, CH2CN, CH2CH2OH, CH2OCH2-phenyl, CH2OH, CO2Me; E1 and E2 may form a ring. SELECTED DRAWING : None COPYRIGHT : (C)2019, JPO&INPIT |
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