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专利概况
专利名称 NOVEL SUBSTITUTED BICYCLIC COMPOUNDS AS BROMODOMAIN INHIBITORS
申请号 JP2018228291 申请日
公开(公告)号 JP2019052178A 公开(公告)日
申请(专利权)人 Zenith Epigenetics Ltd 发明人 LIU SHUANG; JOHN FREDERICK QUINN; BRYAN CORDELL DUFFY; WANG RUIFANG; MAY XIAOWU JIANG; GREGORY SCOTT MARTIN; ZHAO HE; MICHAEL ELLIS; GREGORY STEVEN WAGNER; YOUNG PETER RONALD
专利来源 国家知识产权局 转化方式
摘要

To provide a novel BET protein function inhibitor.SOLUTION : The invention relates to substituted bicyclic compounds, which are useful for inhibition of BET protein function by binding to bromodomains, pharmaceutical compositions comprising these compounds, and use of the compounds and compositions in therapy.SELECTED DRAWING : None

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