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专利概况
专利名称 NEW SALT OF ABEXINOSTAT, ASSOCIATED CRYSTALLINE FORM, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
申请号 JP2018228486 申请日
公开(公告)号 JP2019069955A 公开(公告)日
申请(专利权)人 PHARMACYCLICS LLC 发明人 ANNE PIMONT GARRO; PHILIPPE LETELLIER
专利来源 国家知识产权局 转化方式
摘要

PROBLEM TO BE SOLVED : To provide new salt of abexinostat, associated crystalline form, a process for their preparation and pharmaceutical compositions containing them. SOLUTION : The present invention provides abexinostat tosylate of formula II, and a crystalline form I of the abexinostat tosylate characterized by its powder diffraction pattern X, its Raman spectrum, and its solid 13C CP/MAS NMR spectrum. SELECTED DRAWING : None COPYRIGHT : (C)2019, JPO&INPIT

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