| 专利名称 | NEW SALT OF ABEXINOSTAT, ASSOCIATED CRYSTALLINE FORM, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | ||
| 申请号 | JP2018228486 | 申请日 | |
| 公开(公告)号 | JP2019069955A | 公开(公告)日 | |
| 申请(专利权)人 | PHARMACYCLICS LLC | 发明人 | ANNE PIMONT GARRO; PHILIPPE LETELLIER |
| 专利来源 | 国家知识产权局 | 转化方式 | |
| 摘要 |
PROBLEM TO BE SOLVED : To provide new salt of abexinostat, associated crystalline form, a process for their preparation and pharmaceutical compositions containing them. SOLUTION : The present invention provides abexinostat tosylate of formula II, and a crystalline form I of the abexinostat tosylate characterized by its powder diffraction pattern X, its Raman spectrum, and its solid 13C CP/MAS NMR spectrum. SELECTED DRAWING : None COPYRIGHT : (C)2019, JPO&INPIT |
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