| 专利名称 | BICYCLIC HETEROCYCLES AS FGFR INHIBITORS | ||
| 申请号 | JP2018228352 | 申请日 | |
| 公开(公告)号 | JP2019069953A | 公开(公告)日 | |
| 申请(专利权)人 | INCYTE HOLDINGS CORPORATION | 发明人 | SUN YAPING; LU LIANG; YAO WENQING; ZHUO JINCONG; WU LIANGXING; XU MEIZHONG; QIAN DING QUAN; ZHANG FENGLEI; HE CHUNHONG |
| 专利来源 | 国家知识产权局 | 转化方式 | |
| 摘要 |
PROBLEM TO BE SOLVED : To provide drugs for treatment of cancer and other diseases.SOLUTION : An FGFR inhibitor comprises a formula I or a pharmaceutically acceptable salt thereof. (In the formula, W is NR9 or O; R1 is alkyl; R2 to R5 are H, halo, alkyl, CN, alkoxy, ketone, amide, ester, or the like; R6 is halo, alkyl, CN, NO2, alkoxy, ketone, amide, ester, or the like; and R7 to R9 are H, alkyl, aryl, or the like.)SELECTED DRAWING : NoneCOPYRIGHT : (C)2019, JPO&INPIT |
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