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专利概况
专利名称 MACROCYCLES WITH HETEROCYCLIC P2' GROUPS AS FACTOR XIA INHIBITORS
申请号 JP2019060181 申请日
公开(公告)号 JP2019094354A 公开(公告)日
申请(专利权)人 BRISTOL MYERS SQUIBB COMPANY 发明人 JAMES R CORTE; INDAWATI DLUCCA; FANG TIANAN; YANG WU; WANG YUFENG; ANDREW K DILGER; KUMAR BALASHANMUGA PABBISETTY; WILLIAM R EWING; ZHU YEHENG; RUTH R WEXLER; DONALD J P PINTO; MICHAEL J ORWAT; LEON M SMITH II
专利来源 国家知识产权局 转化方式
摘要

PROBLEM TO BE SOLVED : To provide novel macrocyclic compounds, and analogues (including stereoisomers, tautomers, or pharmaceutically acceptable salts or solvates) thereof, which are useful as selective factor XIa inhibitors or dual inhibitors of factor XIa and plasma kallikrein. SOLUTION : The present invention provides compounds represented by formula (I), where all the variable groups are as defined herein, or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof. These compounds are selective factor XIa inhibitors or dual inhibitors of FXIa and plasma kallikrein. SELECTED DRAWING : None COPYRIGHT : (C)2019, JPO&INPIT

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