专利名称 | USE OF TETRAACETYLATED 5-AMINO-4-CARBAMOYL IMIDAZOLYL-1-β-D-RIBOFURANOSIDE AS A PROTEIN KINASE Cδ INHIBITOR | ||
申请号 | RU2019126467 | 申请日 | |
公开(公告)号 | RU2712150C1 | 公开(公告)日 | |
申请(专利权)人 | OBSHCHESTVO S OGRANICHENNOJ OTVETSTVENNOSTYU TSENTR TRANSFERA BIOTEKHNOLOGIJ OKA BIOTEKH | 发明人 | BEBUROV MIKHAIL YUREVICH; BROVKIN ALEKSEJ NIKOLAEVICH; KALUZHSKIJ VASILIJ EVGENEVICH; LUKYANETS EVGENIJ ANTONOVICH; MAKAROVA ELENA ALEKSANDROVNA; MOSHENTSEVA VERA NIKOLAEVNA; TSVETKOV VLADIMIR BORISOVICH; SHCHERBAKOV ALEKSANDR MIKHAJLOVICH |
专利来源 | 国家知识产权局 | 转化方式 | |
摘要 |
FIELD : chemistry.SUBSTANCE : invention refers to organic chemistry and medicine. Disclosed is use of a tetraacetyled derivative of 5-amino-4-carbamoylimidazolyl-1-β-D-ribofuranoside – ((AcO)4AICAR) as a selective inhibitor of protein kinase Cδ. (AcO)4AICAR effectively inhibits protein kinase Cδ (PKCδ) due to specific inhibition of PKCδ/NF-κB signaling pathway.EFFECT : because (AcO)4AICAR does not possess high toxicity with respect to healthy cells, it allows using it in disturbances prevention of PKCδ/NF-κB signaling pathway, for example to prevent apoptosis or increased thrombosis.4 cl, 4 dwg, 6 ex |
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