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专利概况
专利名称 USE OF TETRAACETYLATED 5-AMINO-4-CARBAMOYL IMIDAZOLYL-1-β-D-RIBOFURANOSIDE AS A PROTEIN KINASE Cδ INHIBITOR
申请号 RU2019126467 申请日
公开(公告)号 RU2712150C1 公开(公告)日
申请(专利权)人 OBSHCHESTVO S OGRANICHENNOJ OTVETSTVENNOSTYU TSENTR TRANSFERA BIOTEKHNOLOGIJ OKA BIOTEKH 发明人 BEBUROV MIKHAIL YUREVICH; BROVKIN ALEKSEJ NIKOLAEVICH; KALUZHSKIJ VASILIJ EVGENEVICH; LUKYANETS EVGENIJ ANTONOVICH; MAKAROVA ELENA ALEKSANDROVNA; MOSHENTSEVA VERA NIKOLAEVNA; TSVETKOV VLADIMIR BORISOVICH; SHCHERBAKOV ALEKSANDR MIKHAJLOVICH
专利来源 国家知识产权局 转化方式
摘要

FIELD : chemistry.SUBSTANCE : invention refers to organic chemistry and medicine. Disclosed is use of a tetraacetyled derivative of 5-amino-4-carbamoylimidazolyl-1-β-D-ribofuranoside – ((AcO)4AICAR) as a selective inhibitor of protein kinase Cδ. (AcO)4AICAR effectively inhibits protein kinase Cδ (PKCδ) due to specific inhibition of PKCδ/NF-κB signaling pathway.EFFECT : because (AcO)4AICAR does not possess high toxicity with respect to healthy cells, it allows using it in disturbances prevention of PKCδ/NF-κB signaling pathway, for example to prevent apoptosis or increased thrombosis.4 cl, 4 dwg, 6 ex

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