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专利概况
专利名称 FUSED PYRIMIDINES AS ISOFORM SELECTIVE PHOSPHOINOSITIDE-3-KINASE-ALPHA INHIBITORS AND PROCESS FOR PREPARATION THEREOF
申请号 US15774520 申请日
公开(公告)号 US20200031845A1 公开(公告)日
申请(专利权)人 Council of Scientific and Industrial Research 发明人 Sandip Bibishan BHARATE; Shashi BHUSHAN; Shabber MOHAMMED; Santosh Kumar GURU; Sonali Sandip BHARATE; Vikas KUMAR; Girish MAHAJAN; Mubashir Javed MINTOO; Dilip Manikrao MONDHE; Ram VISHWAKARMA
专利来源 国家知识产权局 转化方式
摘要

The present invention relates to fused pyrimidines of formulae I and II wherein, R1, R2 are as herein described. The present invention particularly relates to isoform selective PI3Kα inhibition and their medicinal use as anticancer agents.

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