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专利概况
专利名称 CRYSTAL FORM OF SALT OF FUSED TRICYCLIC Γ-AMINO ACID DERIVATIVE AND PREPARATION AND USE THEREOF
申请号 WOCN19095857 申请日
公开(公告)号 WO2020011258A1 公开(公告)日
申请(专利权)人 SICHUAN HAISCO PHARMACEUTICAL CO LTD 发明人 LI Yao; SHI Zongjun; SHI Shaohui; LI Sheng; YAN Pangke; ZHENG Wei
专利来源 国家知识产权局 转化方式
摘要

Provided are a crystal form of a salt of a fused tricyclic γ-amino acid derivative and the preparation and use thereof. As shown in formula (I), Y is selected from maleic acid, fumaric acid, haloid acid (preferably hydrobromic acid and hydrochloric acid), sulfuric acid, phosphoric acid, L-tartaric acid, citric acid, L-malic acid, hippuric acid, D-glucuronic acid, glycollic acid, mucic acid, succinic acid, lactic acid, orotic acid, pamoic acid, malonic acid, gentisic acid, oxalic acid, glutaric acid or saccharin.

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